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Stereoselective syntheses of the trans-decahydroquinoline-5-carboxylic acid epimers. Diastereomeric zwitterionic probes of .gamma.-aminobutyric acid-related biological properties in vitro and in vivo JOURNAL ARTICLE published January 1986 in Journal of Medicinal Chemistry |
Potent angiotensin II antagonists with non-.beta.-branched amino acids in position 5 JOURNAL ARTICLE published February 1989 in Journal of Medicinal Chemistry |
Rigid amino acids related to .alpha.-methyldopa JOURNAL ARTICLE published May 1974 in Journal of Medicinal Chemistry |
Probes for narcotic receptor mediated phenomena. 18. Epimeric 6.alpha.- and 6.beta.-iodo-3,14-dihydroxy-17-(cyclopropylmethyl)-4,5.alpha.-epoxymorphinans as potential ligands for opioid receptor single photon emission computed tomography: synthesis, evaluation, and radiochemistry of [125I]-6.beta.-iodo-3,14-dihydroxy-17-(cyclopropylmethyl)-4,5.alpha.-epoxymorphinan JOURNAL ARTICLE published July 1992 in Journal of Medicinal Chemistry |
Conformational Analysis of Ketolide, Conformations of RU 004 in Solution and Bound to Bacterial Ribosomes JOURNAL ARTICLE published 1 August 1998 in Journal of Medicinal Chemistry |
Synthetic and computer-assisted analyses of the pharmacophore for the benzodiazepine receptor inverse agonist site JOURNAL ARTICLE published September 1990 in Journal of Medicinal Chemistry |
Determining Cysteines Available for Covalent Inhibition Across the Human Kinome JOURNAL ARTICLE published 13 April 2017 in Journal of Medicinal Chemistry Research funded by U.S. National Library of Medicine (R01 LM011986) | National Institute on Minority Health and Health Disparities (G12 MD007599) |
Effects of Bisphosphonates on the Growth of Entamoeba histolytica and Plasmodium Species in Vitro and in Vivo JOURNAL ARTICLE published 1 January 2004 in Journal of Medicinal Chemistry |
Metabolism of 1,3-bis(2-chloroethyl)-1-nitrosourea by rat hepatic microsomes JOURNAL ARTICLE published June 1981 in Journal of Medicinal Chemistry |
The Discovery of Novel Potent trans-3,4-Disubstituted Pyrrolidine Inhibitors of the Human Aspartic Protease Renin from in Silico Three-Dimensional (3D) Pharmacophore Searches JOURNAL ARTICLE published 28 March 2013 in Journal of Medicinal Chemistry |
Design and Synthesis of Brefeldin A Sulfide Derivatives as Prodrug Candidates with Enhanced Aqueous Solubilities JOURNAL ARTICLE published 1 August 1998 in Journal of Medicinal Chemistry |
Bis-cycloSal-d4T-monophosphates: Drugs That Deliver Two Molecules of Bioactive Nucleotides JOURNAL ARTICLE published 1 March 2007 in Journal of Medicinal Chemistry |
Synthesis and Anticonvulsant Activities of (R)-N-(4′-Substituted)benzyl 2-Acetamido-3-methoxypropionamides JOURNAL ARTICLE published 11 February 2010 in Journal of Medicinal Chemistry |
Discovery of Benzocycloalkane Derivatives Efficiently Blocking Bacterial Virulence for the Treatment of Methicillin-Resistant S. aureus (MRSA) Infections by Targeting Diapophytoene Desaturase (CrtN) JOURNAL ARTICLE published 26 May 2016 in Journal of Medicinal Chemistry Research funded by Program for New Century Excellent Talents in University (NCET-12-0853) | Shanghai Municipal Education Commission (14SG28) | National Natural Science Foundation of China (21222211,21372001,21472207) |
Insulin Analogues with Altered Insulin Receptor Isoform Binding Specificities and Enhanced Aggregation Stabilities JOURNAL ARTICLE published 14 October 2021 in Journal of Medicinal Chemistry Research funded by Medical Research Council (MR/K000179/1,MR/R009066/1) | European Regional Development Fund (CZ.02.1.01/0.0/0.0/16_019/0000729) |
Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis JOURNAL ARTICLE published 14 January 2021 in Journal of Medicinal Chemistry |
Issue Editorial Masthead JOURNAL ARTICLE published 11 April 2024 in Journal of Medicinal Chemistry |
Design of Novel 2-Phenylquinazolin-4-amines as Selective CYP1B1 Inhibitors for Overcoming Paclitaxel Resistance in A549 Cells JOURNAL ARTICLE published 11 April 2024 in Journal of Medicinal Chemistry Research funded by National Natural Science Foundation of China (22371026,82001869) | Creative Research Group of CQ University (CXQT21017) | Science and Technology Research Program of Chongqing Municipal Education Commission (KJQN202200446) |
CBP/p300 Degrader: A Promising Therapeutic Strategy for Treatment of Prostate Cancer and Beyond JOURNAL ARTICLE published 11 April 2024 in Journal of Medicinal Chemistry |
Discovery of Near-Infrared Heptamethine Cyanine Probes for Imaging-Guided Surgery in Solid Tumors JOURNAL ARTICLE published 11 April 2024 in Journal of Medicinal Chemistry Research funded by Jiangsu Planned Projects for Postdoctoral Research Funds (2023ZB521) | National Key Research and Development Program of China (2022YFE0138800) | Natural Science Foundation of Jiangsu Province (BE2023842) | Fundamental Research Funds for the Central Universities (2632023GR01) | National Natural Science Foundation of China (82230070) |