Inhibition survey with phenolic compounds against the δ- and η-class carbonic anhydrases from the marine diatom thalassiosira weissflogii and protozoan Plasmodium falciparum

JOURNAL ARTICLE published 1 January 2020 in Journal of Enzyme Inhibition and Medicinal Chemistry

Research funded by Deanship of Scientific Research at Princess Nourah bint Abdulrahman University (RGP-1440–0024)

Authors: Siham A. Alissa | Hanan A. Alghulikah | Zeid A. ALOthman | Sameh M. Osman | Sonia Del Prete | Clemente Capasso | Alessio Nocentini | Claudiu T. Supuran

Molecular engineering of a small trypsin inhibitor based on the binding loop of horsegram seed Bowman-Birk inhibitor

JOURNAL ARTICLE published 1 August 2011 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Deepa G. Muricken | Lalitha R. Gowda

Upcoming conferences of interest

JOURNAL ARTICLE published 1 February 2012 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Claudiu T. Supuran

Synthesis and antiviral activity of 1-(1,3-disubstitutedimidazolidyn-2-ylidene)-3-ethoxycarbonylmethylurea derivatives

JOURNAL ARTICLE published 23 March 2015 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Marzena Rządkowska | Elżbieta Szacoń | Agnieszka A. Kaczor | Barbara Rajtar | Łukasz Świątek | Małgorzata Polz-Dacewicz | Dariusz Matosiuk

Fluorine bearing sydnones with styryl ketone group: synthesis and their possible analgesic and anti-inflammatory activities

JOURNAL ARTICLE published 1 April 2012 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Shreenivas Ramachandrarao Deshpande | Karkala Vasantakumar Pai

N-aryl 2-aryloxyacetamides as a new class of fatty acid amide hydrolase (FAAH) inhibitors

JOURNAL ARTICLE published 1 January 2017 in Journal of Enzyme Inhibition and Medicinal Chemistry

Research funded by Knut och Alice Wallenbergs Stiftelse (2008.0064) | Vetenskapsrådet (521-2012-2802)

Authors: Naresh Sunduru | Mona Svensson | Mariateresa Cipriano | Sania Marwaha | C. David Andersson | Richard Svensson | Christopher J. Fowler | Mikael Elofsson

Synthesis, central nervous system activity and structure–activity relationship of N-substituted derivatives of 1-arylimidazolidyn-2-ylideneurea and products of their cyclization

JOURNAL ARTICLE published 3 September 2015 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Elżbieta Szacoń | Marzena Rządkowska | Agnieszka A. Kaczor | Ewa Kędzierska | Antonina Mazur | Sylwia Fidecka | Dariusz Matosiuk

Ligand design, synthesis and biological anti-HCV evaluations for genotypes 1b and 4a of certain 4-(3- & 4-[3-(3,5-dibromo-4-hydroxyphenyl)-propylamino]phenyl) butyric acids and 3-(3,5-dibromo-4-hydroxyphenyl)-propylamino-acetamidobenzoic acid esters

JOURNAL ARTICLE published 1 December 2013 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Mohamed Abdel Hamid Ismail | Khaled A. M. Abouzid | Nasser Saad Mohamed | Eman Mahmoud Elawady Dokla

Effect of betaine on the hepatic damage from orotic acid-induced fatty liver development in rats

JOURNAL ARTICLE published 13 December 2011 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Jae-Young Cha | Hyeong-Soo Kim | Hyung-In Moon | Young-Su Cho

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

JOURNAL ARTICLE published 1 January 2018 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Giannamaria Annunziato | Laura Giovati | Andrea Angeli | Marialaura Pavone | Sonia Del Prete | Marco Pieroni | Clemente Capasso | Agostino Bruno | Stefania Conti | Walter Magliani | Claudiu T. Supuran | Gabriele Costantino

Studies on synthetic and structural characterization of new fluorine substituted phthalides of pharmaceutical interest

JOURNAL ARTICLE published 1 October 2012 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Tanu Chamoli | M. S. M. Rawat | Melissa Jacob

The effect of some antineoplastic agents on glutathione S-transferase from human erythrocytes

JOURNAL ARTICLE published 1 August 2013 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Mustafa Erat | Halis Şakiroğlu

Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors

JOURNAL ARTICLE published 1 January 2019 in Journal of Enzyme Inhibition and Medicinal Chemistry

Research funded by Regione Autonoma della Sardegna Project L.R. (2012_CRP-59473 to VO) | University of Cagliari (FIR 2016–17) | Swedish Research Council (12158)

Authors: Alessandro Deplano | Mariateresa Cipriano | Federica Moraca | Ettore Novellino | Bruno Catalanotti | Christopher J. Fowler | Valentina Onnis

In vitroeffects of some drugs on human red blood cell glucose-6-phosphate dehydrogenase enzyme activity

JOURNAL ARTICLE published January 2006 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Hasan Özdemir | Mehmet Çiftçi

Anticancer active trifluoromethylated fused triazinones are safe for early-life stages of zebrafish (Danio rerio) and reveal a proapoptotic action

JOURNAL ARTICLE published 1 January 2021 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Małgorzata Sztanke | Jolanta Rzymowska | Krzysztof Sztanke

Novel agonists of free fatty acid receptor 1 (GPR40) based on 3-(1,3,4-thiadiazol-2-yl)propanoic acid scaffold

JOURNAL ARTICLE published 1 November 2016 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Mikhail Krasavin | Alexey Lukin | Nikolay Zhurilo | Alexey Kovalenko | Ihor Zahanich | Sergey Zozulya

Novel diphenyl esters of peptidyl α-aminoalkylphosphonates as inhibitors of chymotrypsin and subtilisin

JOURNAL ARTICLE published 1 December 2009 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Ewa Pietrusewicz | Marcin Sieńczyk | Józef Oleksyszyn

Synthesis of some novel heterocylic compounds derived from 2-[3-(4-chlorophenyl)-5-(4-methoxybenzyl)-4H-1,2,4-triazol-4-yl]acetohydrazide and investigation of their lipase andα-glucosidase inhibition

JOURNAL ARTICLE published 2 November 2015 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: Olcay Bekircan | Serdar Ülker | Emre Menteşe

Correction to: Synthesis, antitumor screening and cell cycle analysis of novel benzothieno[3,2-b]pyran derivatives

JOURNAL ARTICLE published 1 January 2017 in Journal of Enzyme Inhibition and Medicinal Chemistry

Proceedings of the 14^th Annual Conference on the Grouping of Pharmacochemistry of the Atlantic Arc (GP2A)

JOURNAL ARTICLE published 1 January 2006 in Journal of Enzyme Inhibition and Medicinal Chemistry

Authors: G. Le Baut | M. Le Borgne