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Selective Inhibitors of Human Liver Carboxylesterase Based on a β-Lapachone Scaffold: Novel Reagents for Reaction Profiling

JOURNAL ARTICLE published 23 February 2017 in Journal of Medicinal Chemistry

Research funded by National Cancer Institute (CA108775,CA21765) | National Center for Complementary and Integrative Health (AT007531)

Authors: M. Jason Hatfield | Jingwen Chen | Ellie M. Fratt | Liying Chi | John C. Bollinger | Randall J. Binder | John Bowling | Janice L. Hyatt | Jerrod Scarborough | Cynthia Jeffries | Philip M. Potter

https://doi.org/10.1021/acs.jmedchem.6b01849 Actions

Discovery of Targeting Ligands for Breast Cancer Cells Using the One-Bead One-Compound Combinatorial Method

JOURNAL ARTICLE published 8 January 2009 in Journal of Medicinal Chemistry

Authors: Nianhuan Yao | Wenwu Xiao | Xiaobing Wang | Jan Marik | See Hyoung Park | Yoshikazu Takada | Kit S. Lam

https://doi.org/10.1021/jm801062d Actions

Design and Pharmacological Activity of Phosphinic Acid Based NAALADase Inhibitors

JOURNAL ARTICLE published 1 November 2001 in Journal of Medicinal Chemistry

Authors: Paul F. Jackson | Kevin L. Tays | Keith M. Maclin | Yao-Sen Ko | Weixing Li | Dil Vitharana | Takashi Tsukamoto | Doris Stoermer | Xi-Chun M. Lu | Krystyna Wozniak | Barbara S. Slusher

https://doi.org/10.1021/jm0001774 Actions

Sulfamoyl azides. Hydrolysis rates and hypotensive activity

JOURNAL ARTICLE published May 1972 in Journal of Medicinal Chemistry

Authors: W. L. Matier | W. T. Comer | D. Deitchman

https://doi.org/10.1021/jm00275a025 Actions

Solid-Phase Library Synthesis, Screening, and Selection of Tight-Binding Reduced Peptide Bond Inhibitors of a RecombinantLeishmaniamexicanaCysteine Protease B

JOURNAL ARTICLE published 1 May 2002 in Journal of Medicinal Chemistry

Authors: Phaedria M. St. Hilaire | Lira C. Alves | Fatima Herrera | Manat Renil | Sanya J. Sanderson | Jeremy C. Mottram | Graham H. Coombs | Maria A. Juliano | Luiz Juliano | Jorge Arevalo | Morten Meldal

https://doi.org/10.1021/jm0110901 Actions

Structure−Activity Studies of the Melanocortin Peptides:  Discovery of Potent and Selective Affinity Antagonists for thehMC3 andhMC4 Receptors

JOURNAL ARTICLE published 1 November 2002 in Journal of Medicinal Chemistry

Authors: Paolo Grieco | Antonio Lavecchia | Minying Cai | Devendra Trivedi | David Weinberg | Tanya MacNeil | L. H. T. Van der Ploeg | Victor J. Hruby

https://doi.org/10.1021/jm0202526 Actions

Lipoamino Acid-Based Adjuvant Carrier System:  Enhanced Immunogenicity of Group A Streptococcal Peptide Epitopes

JOURNAL ARTICLE published 1 March 2002 in Journal of Medicinal Chemistry

Authors: Anikó Horváth | Colleen Olive | Allan Wong | Timothy Clair | Penny Yarwood | Michael Good | Istvan Toth

https://doi.org/10.1021/jm0110441 Actions

Novel Cyclic Templates of α-MSH Give Highly Selective and Potent Antagonists/Agonists for Human Melanocortin-3/4 Receptors

JOURNAL ARTICLE published 1 June 2002 in Journal of Medicinal Chemistry

Authors: Malcolm J. Kavarana | Dev Trivedi | Minying Cai | Jinfa Ying | Matthew Hammer | Christopher Cabello | Paolo Grieco | Guoxia Han | Victor J. Hruby

https://doi.org/10.1021/jm020021z Actions

Monocyclic Human Tachykinin NK-2 Receptor Antagonists as Evolution of a Potent Bicyclic Antagonist:  QSAR and Site-Directed Mutagenesis Studies

JOURNAL ARTICLE published 1 August 2002 in Journal of Medicinal Chemistry

Authors: Alessandro Giolitti | Maria Altamura | Francesca Bellucci | Danilo Giannotti | Stefania Meini | Riccardo Patacchini | Luigi Rotondaro | Sabrina Zappitelli | Carlo A. Maggi

https://doi.org/10.1021/jm011127h Actions

Synthesis and in Vitro Evaluation of18F- and19F-Labeled Insulin:  A New Radiotracer for PET-based Molecular Imaging Studies

JOURNAL ARTICLE published 1 February 2006 in Journal of Medicinal Chemistry

Authors: Katharina J. Guenther | Sabesan Yoganathan | Robert Garofalo | Thomas Kawabata | Thomas Strack | Renée Labiris | Myrna Dolovich | Raman Chirakal | John F. Valliant

https://doi.org/10.1021/jm0509344 Actions

Procainamide–SAHA Fused Inhibitors of hHDAC6 Tackle Multidrug-Resistant Malaria Parasites

JOURNAL ARTICLE published 22 July 2021 in Journal of Medicinal Chemistry

Research funded by Pasteur Transversal Research Program (PTR 233-2019 HALBY) | Institut Carnot Institut Pasteur (S-CR18089-02B15 DARRI CONSO INNOV 46-19,S-PI15006-10A INNOV 05-2019 ARIMONDO IARP 2019-PC) | Agence national de Recherche (EpiKillMal)

Authors: Flore Nardella | Ludovic Halby | Irina Dobrescu | Johanna Viluma | Corentin Bon | Aurélie Claes | Véronique Cadet-Daniel | Ambre Tafit | Camille Roesch | Elie Hammam | Diane Erdmann | Melissa Mairet-Khedim | Roger Peronet | Salah Mecheri | Benoit Witkowski | Artur Scherf | Paola B. Arimondo

https://doi.org/10.1021/acs.jmedchem.1c00821 Actions

Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines:  Novel Non-Nucleoside Reverse Transcriptase Inhibitors of the S-DABO Series

JOURNAL ARTICLE published 1 May 1997 in Journal of Medicinal Chemistry

Authors: Antonello Mai | Marino Artico | Gianluca Sbardella | Silvana Quartarone | Silvio Massa | Anna G. Loi | Antonella De Montis | Franca Scintu | Monica Putzolu | Paolo La Colla

https://doi.org/10.1021/jm960802y Actions

Synthesis and biological activity of 2'-fluoro-2-halo derivatives of 9-.beta.-D-arabinofuranosyladenine

JOURNAL ARTICLE published January 1992 in Journal of Medicinal Chemistry

Authors: John A. Montgomery | Anita T. Shortnacy-Fowler | Sarah D. Clayton | James M. Riordan | John A. Secrist

https://doi.org/10.1021/jm00080a029 Actions

Novel Tetralone-Derived Retinoic Acid Metabolism Blocking Agents:  Synthesis and in Vitro Evaluation with Liver Microsomal and MCF-7 CYP26A1 Cell Assays

JOURNAL ARTICLE published 1 November 2005 in Journal of Medicinal Chemistry

Authors: Sook Wah Yee | Laetitia Jarno | Mohamed Sayed Gomaa | Carole Elford | Li-Ling Ooi | Michael P. Coogan | Richard McClelland | Robert Ian Nicholson | Bronwen A. J. Evans | Andrea Brancale | Claire Simons

https://doi.org/10.1021/jm0501681 Actions

Second Generation Analogues of the Cancer Drug Clinical Candidate Tipifarnib for Anti-Chagas Disease Drug Discovery

JOURNAL ARTICLE published 27 May 2010 in Journal of Medicinal Chemistry

Authors: James M. Kraus | Hari Babu Tatipaka | Sarah A. McGuffin | Naveen Kumar Chennamaneni | Mandana Karimi | Jenifer Arif | Christophe L. M. J. Verlinde | Frederick S. Buckner | Michael H. Gelb

https://doi.org/10.1021/jm9013136 Actions

Antitumor imidazotetrazines. 25. Crystal structure of 8-carbamoyl-3-methylimidazo[5,1-d]-1,2,3,5-tetrazin-4(3H)-one (temozolomide) and structural comparisons with the related drugs mitozolomide and DTIC

JOURNAL ARTICLE published September 1992 in Journal of Medicinal Chemistry

Authors: P. R. Lowe | C. E. Sansom | C. H. Schwalbe | M. F. G. Stevens | A. S. Clark

https://doi.org/10.1021/jm00096a013 Actions

1,2,5-Thiadizole 1-oxide and 1,1-dioxide derivatives. A new class of potent histamine H2-receptor antagonists

JOURNAL ARTICLE published March 1982 in Journal of Medicinal Chemistry

Authors: Aldo A. Algieri | George M. Luke | Robert T. Standridge | Myron Brown | Richard A. Partyka | R. R. Crenshaw

https://doi.org/10.1021/jm00345a003 Actions

Use of a Pharmacophore Model To Discover a New Class of Influenza Endonuclease Inhibitors

JOURNAL ARTICLE published 1 March 2003 in Journal of Medicinal Chemistry

Authors: Kevin E. B. Parkes | Philipp Ermert | Jürg Fässler | Jane Ives | Joseph A. Martin | John H. Merrett | Daniel Obrecht | Glyn Williams | Klaus Klumpp

https://doi.org/10.1021/jm020334u Actions

5-(Haloalkyl)-2'-deoxyuridines: a novel type of potent antiviral nucleoside analog

JOURNAL ARTICLE published November 1985 in Journal of Medicinal Chemistry

Authors: Herfried Griengl | Michael Bodenteich | Walter Hayden | Erich Wanek | Wolfgang Streicher | Peter Stuetz | Helmut Bachmayer | Ismail Ghazzouli | Brigitte Rosenwirth

https://doi.org/10.1021/jm00149a024 Actions

Discovery of BAY-985, a Highly Selective TBK1/IKKε Inhibitor

JOURNAL ARTICLE published 23 January 2020 in Journal of Medicinal Chemistry

Authors: Julien Lefranc | Volker Klaus Schulze | Roman Christian Hillig | Hans Briem | Florian Prinz | Anne Mengel | Tobias Heinrich | Jozsef Balint | Srinivasan Rengachari | Horst Irlbacher | Detlef Stöckigt | Ulf Bömer | Benjamin Bader | Stefan Nikolaus Gradl | Carl Friedrich Nising | Franz von Nussbaum | Dominik Mumberg | Daniel Panne | Antje Margret Wengner

https://doi.org/10.1021/acs.jmedchem.9b01460 Actions
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