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Selective Inhibitors of Human Liver Carboxylesterase Based on a β-Lapachone Scaffold: Novel Reagents for Reaction Profiling JOURNAL ARTICLE published 23 February 2017 in Journal of Medicinal Chemistry Research funded by National Cancer Institute (CA108775,CA21765) | National Center for Complementary and Integrative Health (AT007531) |
Design and Pharmacological Activity of Phosphinic Acid Based NAALADase Inhibitors JOURNAL ARTICLE published 1 November 2001 in Journal of Medicinal Chemistry |
Solid-Phase Library Synthesis, Screening, and Selection of Tight-Binding Reduced Peptide Bond Inhibitors of a RecombinantLeishmaniamexicanaCysteine Protease B JOURNAL ARTICLE published 1 May 2002 in Journal of Medicinal Chemistry |
Novel Cyclic Templates of α-MSH Give Highly Selective and Potent Antagonists/Agonists for Human Melanocortin-3/4 Receptors JOURNAL ARTICLE published 1 June 2002 in Journal of Medicinal Chemistry |
Monocyclic Human Tachykinin NK-2 Receptor Antagonists as Evolution of a Potent Bicyclic Antagonist: QSAR and Site-Directed Mutagenesis Studies JOURNAL ARTICLE published 1 August 2002 in Journal of Medicinal Chemistry |
Synthesis and in Vitro Evaluation of18F- and19F-Labeled Insulin: A New Radiotracer for PET-based Molecular Imaging Studies JOURNAL ARTICLE published 1 February 2006 in Journal of Medicinal Chemistry |
Procainamide–SAHA Fused Inhibitors of hHDAC6 Tackle Multidrug-Resistant Malaria Parasites JOURNAL ARTICLE published 22 July 2021 in Journal of Medicinal Chemistry Research funded by Pasteur Transversal Research Program (PTR 233-2019 HALBY) | Institut Carnot Institut Pasteur (S-CR18089-02B15 DARRI CONSO INNOV 46-19,S-PI15006-10A INNOV 05-2019 ARIMONDO IARP 2019-PC) | Agence national de Recherche (EpiKillMal) |
Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines: Novel Non-Nucleoside Reverse Transcriptase Inhibitors of the S-DABO Series JOURNAL ARTICLE published 1 May 1997 in Journal of Medicinal Chemistry |
Novel Tetralone-Derived Retinoic Acid Metabolism Blocking Agents: Synthesis and in Vitro Evaluation with Liver Microsomal and MCF-7 CYP26A1 Cell Assays JOURNAL ARTICLE published 1 November 2005 in Journal of Medicinal Chemistry |
Antitumor imidazotetrazines. 25. Crystal structure of 8-carbamoyl-3-methylimidazo[5,1-d]-1,2,3,5-tetrazin-4(3H)-one (temozolomide) and structural comparisons with the related drugs mitozolomide and DTIC JOURNAL ARTICLE published September 1992 in Journal of Medicinal Chemistry |
1,2,5-Thiadizole 1-oxide and 1,1-dioxide derivatives. A new class of potent histamine H2-receptor antagonists JOURNAL ARTICLE published March 1982 in Journal of Medicinal Chemistry |
5-(Haloalkyl)-2'-deoxyuridines: a novel type of potent antiviral nucleoside analog JOURNAL ARTICLE published November 1985 in Journal of Medicinal Chemistry |
Discovery of BAY-985, a Highly Selective TBK1/IKKε Inhibitor JOURNAL ARTICLE published 23 January 2020 in Journal of Medicinal Chemistry |
5-C-Branched Deoxynojirimycin: Strategy for Designing a 1-Deoxynojirimycin-Based Pharmacological Chaperone with a Nanomolar Affinity for Pompe Disease JOURNAL ARTICLE published 10 February 2022 in Journal of Medicinal Chemistry Research funded by Japan Society for the Promotion of Science (JP21K06451) | National Natural Science Foundation of China (21272240) |
Development of a 1,2,4-Triazole-Based Lead Tankyrase Inhibitor: Part II JOURNAL ARTICLE published 23 December 2021 in Journal of Medicinal Chemistry Research funded by Norges Forskningsr??d (262613,267639) | Academy of Finland (287063,294085,319299) | South-Eastern Norway Regional Health Authority (15/00779-2,16/00528-9,2015012,2019090,2021035) |
Synthesis and Cytotoxic Evaluation of Combretafurans, Potential Scaffolds for Dual-Action Antitumoral Agents JOURNAL ARTICLE published 1 August 2006 in Journal of Medicinal Chemistry |
Synthesis and Characterization of a Novel Gadolinium-Based Contrast Agent for Magnetic Resonance Imaging of Myelination JOURNAL ARTICLE published 28 February 2013 in Journal of Medicinal Chemistry |
Nitric Oxide Synthase Inhibitors That Interact with Both Heme Propionate and Tetrahydrobiopterin Show High Isoform Selectivity JOURNAL ARTICLE published 22 May 2014 in Journal of Medicinal Chemistry Research funded by National Institutes of Health (GM049725) |
7-Deazaadenines Bearing Polar Substituents: Structure−Activity Relationships of New A1 and A3 Adenosine Receptor Antagonists JOURNAL ARTICLE published 1 November 2000 in Journal of Medicinal Chemistry |
Application of the λ-Dynamics Method To Evaluate the Relative Binding Free Energies of Inhibitors to HCV Protease JOURNAL ARTICLE published 1 December 2003 in Journal of Medicinal Chemistry |