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Design and synthesis of 3,7-diarylimidazopyridines as inhibitors of the VEGF-receptor KDR

JOURNAL ARTICLE published February 2004 in Bioorganic & Medicinal Chemistry Letters

Authors: Zhicai Wu | Mark E. Fraley | Mark T. Bilodeau | Mildred L. Kaufman | Edward S. Tasber | Adrienne E. Balitza | George D. Hartman | Kathleen E. Coll | Keith Rickert | Jennifer Shipman | Bin Shi | Laura Sepp-Lorenzino | Kenneth A. Thomas

Synthesis and biological evaluation of new glutamic acid-based inhibitors of MurD ligase

JOURNAL ARTICLE published January 2009 in Bioorganic & Medicinal Chemistry Letters

Authors: Tihomir Tomašić | Nace Zidar | Veronika Rupnik | Andreja Kovač | Didier Blanot | Stanislav Gobec | Danijel Kikelj | Lucija Peterlin Mašič

N -Alkylaminoacids and Their derivatives interact with melanocortin receptors

JOURNAL ARTICLE published April 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Felikss Mutulis | Ilze Mutule | Jarl E.S. Wikberg

Synthesis and biological evaluation of retinoid-chalcones as inhibitors of colon cancer cell growth

JOURNAL ARTICLE published December 2010 in Bioorganic & Medicinal Chemistry Letters

Authors: Cassia S. Mizuno | Shiby Paul | Nanjoo Suh | Agnes M. Rimando

Discovery of phenyl alanine derived ketoamides carrying benzoyl residues as novel calpain inhibitors

JOURNAL ARTICLE published May 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: W. Lubisch | A. Möller

Stereoselective Synthesis of Ψ[CH 2 O] Pseudodipeptides and Conformational Analysis of a PheΨ[CH 2 O]Ala Containing Analogue of the Drug Desmopressin

JOURNAL ARTICLE published March 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Mattias Hedenström | Lotta Holm | ZhongQing Yuan | Hans Emtenäs | Jan Kihlberg

Synthesis and evaluation of vancomycin and vancomycin aglycon analogues that bear modifications in the residue 3 asparagine

JOURNAL ARTICLE published May 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: J.Jeffrey McAtee | Steven L Castle | Qing Jin | Dale L Boger

Syntheses of Polycationic Dendrimers on Lipophilic Peptide Core for Complexation and Transport of Oligonucleotides

JOURNAL ARTICLE published September 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Norbert Wimmer | Robert J. Marano | Philip S. Kearns | Elizabeth P. Rakoczy | Istvan Toth

Bivalent inhibition of β-Tryptase: distance scan of neighboring subunits by dibasic inhibitors

JOURNAL ARTICLE published March 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Norbert Schaschke | Andreas Dominik | Gabriele Matschiner | Christian P. Sommerhoff

First and unexpected synthesis of macrocyclic cyclophane-based unusual α-amino acid derivatives by phosphazene base without high dilution conditions

JOURNAL ARTICLE published April 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Sambasivarao Kotha | Somnath Halder | Lakshminarasimhan Damodharan | Vasantha Pattabhi

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: Substitution of the glycine part

JOURNAL ARTICLE published October 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Katie Amssoms | Sandra L Oza | Koen Augustyns | Abdellah Yamani | Anne-Marie Lambeir | Gunther Bal | Pieter Van der Veken | Alan H Fairlamb | Achiel Haemers

Solid-phase synthesis of dual α4β1/α4β7 integrin antagonists: two scaffolds with overlapping pharmacophores

JOURNAL ARTICLE published October 2002 in Bioorganic & Medicinal Chemistry Letters

Authors: Georgette M. Castanedo | Fredrick C. Sailes | Nathan J.P. Dubree | John B. Nicholas | Lisa Caris | Kevin Clark | Susan M. Keating | Maureen H. Beresini | Henry Chiu | Sherman Fong | James C. Marsters | David Y. Jackson | Daniel P. Sutherlin

Enzymatic synthesis of aza-l-tyrosines

JOURNAL ARTICLE published August 2001 in Bioorganic & Medicinal Chemistry Letters

Authors: E.Blake Watkins | Robert S Phillips

Antioxidative oligostilbenes from Caragana sinica

JOURNAL ARTICLE published January 2012 in Bioorganic & Medicinal Chemistry Letters

Authors: Qinghao Jin | Xiang Hua Han | Seong Su Hong | Chul Lee | Sanggil Choe | Dongho Lee | Youngsoo Kim | Jin Tae Hong | Mi Kyeong Lee | Bang Yeon Hwang

Synthesis and antimicrobial activity of some new pyrazole derivatives containing a ferrocene unit

JOURNAL ARTICLE published February 2009 in Bioorganic & Medicinal Chemistry Letters

Authors: Ivan Damljanović | Mirjana Vukićević | Niko Radulović | Radosav Palić | Ernst Ellmerer | Zoran Ratković | Milan D. Joksović | Rastko D. Vukićević

Synthesis and evaluation of diacylhydrazines as inhibitors of the interleukin-1β converting enzyme (ICE)

JOURNAL ARTICLE published June 1995 in Bioorganic & Medicinal Chemistry Letters

Authors: Todd L. Graybill | Roland E. Dolle | Carla T. Helaszek | Mark A. Ator | Joost Strasters

Synthesis and evaluation of tricyclic pyrrolopyrimidinones as dipeptide mimetics: Inhibition of interleukin-1β-converting enzyme

JOURNAL ARTICLE published October 2005 in Bioorganic & Medicinal Chemistry Letters

Authors: Michael C. Laufersweiler | Yili Wang | David L. Soper | Maureen K. Suchanek | Amy N. Fancher | Wei Lu | Richard L. Wang | Kofi A. Oppong | Christopher D. Ellis | Mark W. Baize | Steven V. O’Neil | John A. Wos | Thomas P. Demuth

Substituted diaryl ether compounds as retinoic acid-related orphan Receptor-γt (RORγt) agonists

JOURNAL ARTICLE published March 2021 in Bioorganic & Medicinal Chemistry Letters

Authors: Zheming Ruan | Peter K. Park | Donna Wei | Ashok Purandare | Honghe Wan | Daniel O'Malley | Sylwia Stachura | Heidi Perez | Cullen L. Cavallaro | Carolyn A. Weigelt | John S. Sack | Max Ruzanov | Javed Khan | Murali Gururajan | Jessica J. Wong | Yanling Huang | Melissa Yarde | Zhuyin Li | Cliff Chen | Huadong Sun | Virna Borowski | Jenny H. Xie | Monique Anthony | Michele Agler | Brian E. Fink | Lalgudi S. Harikrishnan

Oxamyl dipeptide caspase inhibitors developed for the treatment of stroke

JOURNAL ARTICLE published May 2004 in Bioorganic & Medicinal Chemistry Letters

Authors: Steven D. Linton | Teresa Aja | Peter R. Allegrini | Thomas L. Deckwerth | Jose-Luis Diaz | Bastian Hengerer | Julia Herrmann | Kathy G. Jahangiri | Joerg Kallen | Donald S. Karanewsky | Steven P. Meduna | Kip Nalley | Edward D. Robinson | Silvio Roggo | Giorgio Rovelli | Andre Sauter | Robert O. Sayers | Albert Schmitz | Robert Smidt | Robert J. Ternansky | Kevin J. Tomaselli | Brett R. Ullman | Christoph Wiessner | Joe C. Wu

In situ generated O-Glycan core 1 structure as substrate for Gal(β1–3)GalNAc β-1,6-GlcNAc Transferase

JOURNAL ARTICLE published September 1998 in Bioorganic & Medicinal Chemistry Letters

Authors: Gregor Dudziak | Steffen Zeng | Eric G. Berger | Ricardo Gutiérrez Gallego | Johannis P. Kamerling | Udo Kragl | Christian Wandrey