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Showing results for ISSN matching 0022-2623

Phosphate Chemical Probes Designed for Location Specific Inhibition of Intracellular Carbonic Anhydrases

JOURNAL ARTICLE published 24 September 2015 in Journal of Medicinal Chemistry

Research funded by Australian Research Council (DP110100071,FT10100185)

Authors: Gregory M. Rankin | Daniela Vullo | Claudiu T. Supuran | Sally-Ann Poulsen

https://doi.org/10.1021/acs.jmedchem.5b01228 Actions

Exploration of the Amine Terminus in a Novel Series of 1,2,4-Triazolo-3-yl-azabicyclo[3.1.0]hexanes as Selective Dopamine D3 Receptor Antagonists

JOURNAL ARTICLE published 14 October 2010 in Journal of Medicinal Chemistry

Authors: Fabrizio Micheli | Luca Arista | Barbara Bertani | Simone Braggio | Anna Maria Capelli | Susanna Cremonesi | Romano Di-Fabio | Giacomo Gelardi | Gabriella Gentile | Carla Marchioro | Alessandra Pasquarello | Stefano Provera | Giovanna Tedesco | Luca Tarsi | Silvia Terreni | Angela Worby | Christian Heidbreder

https://doi.org/10.1021/jm100832d Actions

Structure−Activity Studies on a Series of a 2-Aminopyrimidine-Containing Histamine H4 Receptor Ligands

JOURNAL ARTICLE published 23 October 2008 in Journal of Medicinal Chemistry

Authors: Robert J. Altenbach | Ronald M. Adair | Brian M. Bettencourt | Lawrence A. Black | Shannon R. Fix-Stenzel | Sujatha M. Gopalakrishnan | Gin C. Hsieh | Huaqing Liu | Kennan C. Marsh | Michael J. McPherson | Ivan Milicic | Thomas R. Miller | Timothy A. Vortherms | Usha Warrior | Jill M. Wetter | Neil Wishart | David G. Witte | Prisca Honore | Timothy A. Esbenshade | Arthur A. Hancock | Jorge D. Brioni | Marlon D. Cowart

https://doi.org/10.1021/jm8005959 Actions

Quick Assembly of 1,4-Diphenyltriazoles as Probes Targeting β-Amyloid Aggregates in Alzheimer's Disease

JOURNAL ARTICLE published 1 July 2007 in Journal of Medicinal Chemistry

Authors: Wenchao Qu | Mei-Ping Kung | Catherine Hou | Shunichi Oya | Hank F. Kung

https://doi.org/10.1021/jm070467l Actions

Molecular Determinants of MAO Selectivity in a Series of Indolylmethylamine Derivatives:  Biological Activities, 3D-QSAR/CoMFA Analysis, and Computational Simulation of Ligand Recognition

JOURNAL ARTICLE published 1 May 2000 in Journal of Medicinal Chemistry

Authors: Jose A. Morón | Mercedes Campillo | Virgili Perez | Mercedes Unzeta | Leonardo Pardo

https://doi.org/10.1021/jm991164x Actions

Comparative cytotoxic and biochemical effects of ligands and metal complexes of .alpha.-N-heterocyclic carboxaldehyde thiosemicarbazones

JOURNAL ARTICLE published October 1979 in Journal of Medicinal Chemistry

Authors: Leon A. Saryan | Else Ankel | Chitra Krishnamurti | David H. Petering | Howard Elford

https://doi.org/10.1021/jm00196a013 Actions

Optical resolution, absolute configuration, and activity of the enantiomers of proxyphylline

JOURNAL ARTICLE published October 1983 in Journal of Medicinal Chemistry

Authors: Kirsten Selvig | Merete Ruud-Christensen | Arne J. Aasen

https://doi.org/10.1021/jm00364a029 Actions

NO-Donor COX-2 Inhibitors. New Nitrooxy-Substituted 1,5-Diarylimidazoles Endowed with COX-2 Inhibitory and Vasodilator Properties

JOURNAL ARTICLE published 1 April 2007 in Journal of Medicinal Chemistry

Authors: Konstantin Chegaev | Loretta Lazzarato | Paolo Tosco | Clara Cena | Elisabetta Marini | Barbara Rolando | Pierre-Alain Carrupt | Roberta Fruttero | Alberto Gasco

https://doi.org/10.1021/jm0607247 Actions

Synthesis and Optimization of a New Family of Type 3 17β-Hydroxysteroid Dehydrogenase Inhibitors by Parallel Liquid-Phase Chemistry

JOURNAL ARTICLE published 1 January 2002 in Journal of Medicinal Chemistry

Authors: René Maltais | Van Luu-The | Donald Poirier

https://doi.org/10.1021/jm010286y Actions

Corrections to Rational Modification of a Candidate Cancer Drug for Use against Chagas Disease

JOURNAL ARTICLE published 23 July 2009 in Journal of Medicinal Chemistry

Authors: James M. Kraus | Christophe L. M. J. Verlinde | Mandana Karimi | Galina I. Lepesheva | Michael H. Gelb | Frederick S. Buckner

https://doi.org/10.1021/jm900650s Actions

Structure Based Development of Phenylimidazole-Derived Inhibitors of Indoleamine 2,3-Dioxygenase

JOURNAL ARTICLE published 1 August 2008 in Journal of Medicinal Chemistry

Authors: Sanjeev Kumar | Daniel Jaller | Bhumika Patel | Judith M. LaLonde | James B. DuHadaway | William P. Malachowski | George C. Prendergast | Alexander J. Muller

https://doi.org/10.1021/jm800512z Actions

New Anticancer Agents Mimicking Protein Recognition Motifs

JOURNAL ARTICLE published 12 September 2013 in Journal of Medicinal Chemistry

Authors: Marco Persico | Anna Ramunno | Vita Maglio | Silvia Franceschelli | Chiara Esposito | Alfonso Carotenuto | Diego Brancaccio | Valeria De Pasquale | Luigi Michele Pavone | Michela Varra | Nausicaa Orteca | Ettore Novellino | Caterina Fattorusso

https://doi.org/10.1021/jm400947b Actions

Synthesis of two metabolites of (+)-propoxyphene

JOURNAL ARTICLE published August 1977 in Journal of Medicinal Chemistry

Authors: William W. Turner | Richard N. Booher | Stephen E. Smits | Albert Pohland

https://doi.org/10.1021/jm00218a015 Actions

Miliusanes, A Class of Cytotoxic Agents from Miliusa sinensis

JOURNAL ARTICLE published 1 January 2006 in Journal of Medicinal Chemistry

Authors: Hong-Jie Zhang | Cuiying Ma | Nguyen Van Hung | Nguyen Manh Cuong | Ghee Teng Tan | Bernard D. Santarsiero | Andrew D. Mesecar | D. Doel Soejarto | John M. Pezzuto | Harry H. S. Fong

https://doi.org/10.1021/jm0509492 Actions

Acridine-Based Agents with Topoisomerase II Activity Inhibit Pancreatic Cancer Cell Proliferation and Induce Apoptosis

JOURNAL ARTICLE published 1 January 2008 in Journal of Medicinal Chemistry

Authors: John R. Goodell | Andrei V. Ougolkov | Hiroshi Hiasa | Harneet Kaur | Rory Remmel | Daniel D. Billadeau | David M. Ferguson

https://doi.org/10.1021/jm701228e Actions

Targeting Carnitine Biosynthesis: Discovery of New Inhibitors against γ-Butyrobetaine Hydroxylase

JOURNAL ARTICLE published 27 March 2014 in Journal of Medicinal Chemistry

Authors: Kaspars Tars | Janis Leitans | Andris Kazaks | Diana Zelencova | Edgars Liepinsh | Janis Kuka | Marina Makrecka | Daina Lola | Viktors Andrianovs | Daina Gustina | Solveiga Grinberga | Edvards Liepinsh | Ivars Kalvinsh | Maija Dambrova | Einars Loza | Osvalds Pugovics

https://doi.org/10.1021/jm401603e Actions

Structure−Selectivity Investigations of D2-Like Receptor Ligands by CoMFA and CoMSIA Guiding the Discovery of D3Selective PET Radioligands

JOURNAL ARTICLE published 8 February 2007 in Journal of Medicinal Chemistry

Authors: Ismail Salama | Carsten Hocke | Wolfgang Utz | Olaf Prante | Frank Boeckler | Harald Hübner | Torsten Kuwert | Peter Gmeiner

https://doi.org/10.1021/jm0611152 Actions

2,6,8-Trisubstituted 1-Deazapurines as Adenosine Receptor Antagonists

JOURNAL ARTICLE published 1 February 2007 in Journal of Medicinal Chemistry

Authors: Lisa C. W. Chang | Jacobien K. von Frijtag Drabbe Künzel | Thea Mulder-Krieger | Joost Westerhout | Thomas Spangenberg | Johannes Brussee | Adriaan P. IJzerman

https://doi.org/10.1021/jm0607956 Actions

Design, Synthesis, Structure−Selectivity Relationship, and Effect on Human Cancer Cells of a Novel Series of Histone Deacetylase 6-Selective Inhibitors

JOURNAL ARTICLE published 1 November 2007 in Journal of Medicinal Chemistry

Authors: Yukihiro Itoh | Takayoshi Suzuki | Akiyasu Kouketsu | Nobuaki Suzuki | Satoko Maeda | Minoru Yoshida | Hidehiko Nakagawa | Naoki Miyata

https://doi.org/10.1021/jm7009217 Actions

Modeling, Chemistry, and Biology of the Benzolactam Analogues of Indolactam V (ILV). 2. Identification of the Binding Site of the Benzolactams in the CRD2 Activator-Binding Domain of PKCδ and Discovery of an ILV Analogue of Improved Isozyme Selectivity

JOURNAL ARTICLE published 1 April 1997 in Journal of Medicinal Chemistry

Authors: Alan P. Kozikowski | Shaomeng Wang | Dawei Ma | Jiangchao Yao | Shakeel Ahmad | Robert I. Glazer | Krisztina Bogi | Peter Acs | Shayan Modarres | Nancy E. Lewin | Peter M. Blumberg

https://doi.org/10.1021/jm960875h Actions
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