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Showing results for ISSN matching 0022-2623

Preventive Oral Treatment with Resveratrol Pro-prodrugs Drastically Reduce Colon Inflammation in Rodents

JOURNAL ARTICLE published 28 October 2010 in Journal of Medicinal Chemistry

Authors: Mar Larrosa | Joao Tomé-Carneiro | María J. Yáñez-Gascón | David Alcántara | María V. Selma | David Beltrán | María T. García-Conesa | Cristina Urbán | Ricardo Lucas | Francisco Tomás-Barberán | Juan C. Morales | Juan Carlos Espín

https://doi.org/10.1021/jm1007006 Actions

Design, Synthesis, and Biological Evaluation of Monopyrrolinone-Based HIV-1 Protease Inhibitors

JOURNAL ARTICLE published 1 May 2003 in Journal of Medicinal Chemistry

Authors: Amos B. Smith | Louis-David Cantin | Alexander Pasternak | Lisa Guise-Zawacki | Wenquin Yao | Adam K. Charnley | Joseph Barbosa | Paul A. Sprengeler | Ralph Hirschmann | Sanjeev Munshi | David B. Olsen | William A. Schleif | Lawrence C. Kuo

https://doi.org/10.1021/jm0204587 Actions

Development of Novel Aminoglycoside (NB54) with Reduced Toxicity and Enhanced Suppression of Disease-Causing Premature Stop Mutations

JOURNAL ARTICLE published 14 May 2009 in Journal of Medicinal Chemistry

Authors: Igor Nudelman | Annie Rebibo-Sabbah | Marina Cherniavsky | Valery Belakhov | Mariana Hainrichson | Fuquan Chen | Jochen Schacht | Daniel S. Pilch | Tamar Ben-Yosef | Timor Baasov

https://doi.org/10.1021/jm801640k Actions

Design, Synthesis, and Antiviral Activity of Certain 2,5,6-Trihalo-1-(.beta.-D-ribofuranosyl)benzimidazoles

JOURNAL ARTICLE published September 1995 in Journal of Medicinal Chemistry

Authors: Leroy B. Townsend | Rodrigo V. Devivar | Steven R. Turk | M. Reza Nassiri | John C. Drach

https://doi.org/10.1021/jm00020a025 Actions

Synthesis and Anticancer Activity of Brefeldin A Ester Derivatives

JOURNAL ARTICLE published 1 June 2006 in Journal of Medicinal Chemistry

Authors: Nwanne O. Anadu | V. Jo Davisson | Mark Cushman

https://doi.org/10.1021/jm0602817 Actions

Structure−Activity Relationships of New 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as Allosteric Enhancers of the A3 Adenosine Receptor

JOURNAL ARTICLE published 1 June 2006 in Journal of Medicinal Chemistry

Authors: Anikó Göblyös | Zhan-Guo Gao | Johannes Brussee | Roberto Connestari | Sabrina Neves Santiago | Kai Ye | Adriaan P. IJzerman | Kenneth A. Jacobson

https://doi.org/10.1021/jm060086s Actions

Synthesis and Antiprotozoal Activity of N-Alkoxy Analogues of the Trypanocidal Lead Compound 4,4′-Bis(imidazolinylamino)diphenylamine with Improved Human Blood−Brain Barrier Permeability

JOURNAL ARTICLE published 27 January 2011 in Journal of Medicinal Chemistry

Authors: Lidia Nieto | Ainhoa Mascaraque | Florence Miller | Fabienne Glacial | Carlos Ríos Martínez | Marcel Kaiser | Reto Brun | Christophe Dardonville

https://doi.org/10.1021/jm101335q Actions

Enzyme-Activated Antagonists of the Strychnine-Insensitive Glycine/NMDA Receptor

JOURNAL ARTICLE published February 1994 in Journal of Medicinal Chemistry

Authors: Francesco G. Salituro | Ronald C. Tomlinson | Bruce M. Baron | Michael G. Palfreyman | Ian A. McDonald | Werner Schmidt | Hui Qiu Wu | Paolo Guidetti | Robert Schwarcz

https://doi.org/10.1021/jm00029a003 Actions

Synthesis and Characterization of an A6-A11 Methylene Thioacetal Human Insulin Analogue with Enhanced Stability

JOURNAL ARTICLE published 26 December 2019 in Journal of Medicinal Chemistry

Research funded by American Diabetes Association (#1-19-PDF110) | National Institute of Diabetes and Digestive and Kidney Diseases (R01DK120430)

Authors: Nan Zheng | Prasoona Karra | Michael A. VandenBerg | Jin Hwan Kim | Matthew J. Webber | William L. Holland | Danny Hung-Chieh Chou

https://doi.org/10.1021/acs.jmedchem.9b01589 Actions

Synthesis of (E)-5-(3,3,3-trifluoro-1-propenyl)-2'-deoxyuridine and related analogs: potent and unusually selective antiviral activity of (E)-5-(3,3,3-trifluoro-1-propenyl)-2'-deoxyridine against herpes simplex virus type 1

JOURNAL ARTICLE published March 1984 in Journal of Medicinal Chemistry

Authors: Donald E. Bergstrom | Jerry L. Ruth | P. Anantha Reddy | Erik De Clercq

https://doi.org/10.1021/jm00369a009 Actions

Novel Synthesis and Structural Characterization of a High-Affinity Paramagnetic Kinase Probe for the Identification of Non-ATP Site Binders by Nuclear Magnetic Resonance

JOURNAL ARTICLE published 11 February 2010 in Journal of Medicinal Chemistry

Authors: Franklin J. Moy | Arthur Lee | Lori Krim Gavrin | Zhang Bao Xu | Annette Sievers | Elizabeth Kieras | Wayne Stochaj | Lidia Mosyak | John McKew | Désirée H. H. Tsao

https://doi.org/10.1021/jm901525b Actions

Structure-Based Design, Synthesis, Evaluation, and Crystallographic Studies of Conformationally Constrained Smac Mimetics as Inhibitors of the X-linked Inhibitor of Apoptosis Protein (XIAP)

JOURNAL ARTICLE published 27 November 2008 in Journal of Medicinal Chemistry

Authors: Haiying Sun | Jeanne A. Stuckey | Zaneta Nikolovska-Coleska | Dongguang Qin | Jennifer L. Meagher | Su Qiu | Jianfeng Lu | Chao-Yie Yang | Naoyuki G. Saito | Shaomeng Wang

https://doi.org/10.1021/jm8006849 Actions

Effect of Chiral Purity on Adjuvanticity of Archaeol-Based Glycolipids

JOURNAL ARTICLE published 23 June 2022 in Journal of Medicinal Chemistry

Authors: Sophie Régnier | Edmond Lam | Vinicio Vasquez | Camilo F. Martinez-Farina | Felicity C. Stark | Gerard Agbayani | Lise Deschatelets | Renu Dudani | Blair A. Harrison | Bassel Akache | Michael J. McCluskie | Usha D. Hemraz

https://doi.org/10.1021/acs.jmedchem.2c00072 Actions

2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 1. Identification of an Allosteric Binding Site

JOURNAL ARTICLE published 28 February 2019 in Journal of Medicinal Chemistry

Research funded by Deutsche Forschungsgemeinschaft (EN381/2-3) | R?gion Rh?ne-Alpes (?ARC 1 Sant?? 12-008707-01)

Authors: Benoît Bestgen | Isabelle Krimm | Irina Kufareva | Ahmed Ashraf Moustafa Kamal | Wei-Guang Seetoh | Chris Abell | Rolf W. Hartmann | Ruben Abagyan | Claude Cochet | Marc Le Borgne | Matthias Engel | Thierry Lomberget

https://doi.org/10.1021/acs.jmedchem.8b01766 Actions

Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrimido[5,4-b]pyrrolizines as Novel Bruton’s Tyrosine Kinase Inhibitors

JOURNAL ARTICLE published 24 May 2018 in Journal of Medicinal Chemistry

Research funded by Government of Jiangsu Province (KYCX17_0684) | Science and Technology Commission of Shanghai Municipality (16XD1404600,14431900400) | National Natural Science Foundation of China (81703327,81773565,81430080) | Chinese Academy of Sciences (160621,GJHZ1622)

Authors: Yu Xue | Peiran Song | Zilan Song | Aoli Wang | Linjiang Tong | Meiyu Geng | Jian Ding | Qingsong Liu | Liping Sun | Hua Xie | Ao Zhang

https://doi.org/10.1021/acs.jmedchem.8b00441 Actions

Synthesis and Anticonvulsant Activity of Amino Acid-Derived Sulfamides

JOURNAL ARTICLE published 26 March 2009 in Journal of Medicinal Chemistry

Authors: Luciana Gavernet | Juan E. Elvira | Gisela A. Samaja | Valentina Pastore | Mariana Sella Cravero | Andrea Enrique | Guillermina Estiu | Luis E. Bruno-Blanch

https://doi.org/10.1021/jm800764p Actions

Subtype Selective Substrates for Histone Deacetylases

JOURNAL ARTICLE published 1 October 2004 in Journal of Medicinal Chemistry

Authors: Birgit Heltweg | Franck Dequiedt | Brett L. Marshall | Carsten Brauch | Minoru Yoshida | Norikazu Nishino | Eric Verdin | Manfred Jung

https://doi.org/10.1021/jm0497592 Actions

Synthesis, Structure−Activity Relationships, and Characterization of Novel Nonsteroidal and Selective Androgen Receptor Modulators

JOURNAL ARTICLE published 26 November 2009 in Journal of Medicinal Chemistry

Authors: Nathalie Schlienger | Birgitte W. Lund | Jan Pawlas | Fabrizio Badalassi | Fabio Bertozzi | Rasmus Lewinsky | Alma Fejzic | Mikkel B. Thygesen | Ali Tabatabaei | Stefania Risso Bradley | Luis R. Gardell | Fabrice Piu | Roger Olsson

https://doi.org/10.1021/jm901149c Actions

A Straightforward Approach for Engineering Efficacy and Selectivity at GPCRs

JOURNAL ARTICLE published 9 August 2012 in Journal of Medicinal Chemistry

Authors: Stefania Butini | Sandra Gemma | Giuseppe Campiani

https://doi.org/10.1021/jm301017v Actions

Issue Editorial Masthead

JOURNAL ARTICLE published 28 February 2019 in Journal of Medicinal Chemistry

https://doi.org/10.1021/jmv062i004_1261123 Actions
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