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Spirocyclic β-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors: From Hit to Lowering of Cerebrospinal Fluid (CSF) Amyloid β in a Higher Species JOURNAL ARTICLE published 25 April 2013 in Journal of Medicinal Chemistry |
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Synthesis of Cytotoxic 6E-Hydroximino-4-ene Steroids: Structure/Activity Studies JOURNAL ARTICLE published 1 August 2001 in Journal of Medicinal Chemistry |
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Design, Synthesis, and Inhibitory Activity of Potent, Photoswitchable Mast Cell Activation Inhibitors JOURNAL ARTICLE published 13 June 2013 in Journal of Medicinal Chemistry |
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Piperidino Groups in Antitussive Activity JOURNAL ARTICLE published March 1963 in Journal of Medicinal Chemistry |
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Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 2. Selective and Potent Benzylamino Cyclobutenediones JOURNAL ARTICLE published 1 March 2000 in Journal of Medicinal Chemistry |
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First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling JOURNAL ARTICLE published 1 January 2003 in Journal of Medicinal Chemistry |
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Modeling Cyclooxygenase Inhibition. Implication of Active Site Hydration on the Selectivity of Ketoprofen Analogues JOURNAL ARTICLE published 1 June 2000 in Journal of Medicinal Chemistry |
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Study on Affinity Profile toward Native Human and Bovine Adenosine Receptors of a Series of 1,8-Naphthyridine Derivatives JOURNAL ARTICLE published 1 June 2004 in Journal of Medicinal Chemistry |
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Diarylureas as Allosteric Modulators of the Cannabinoid CB1 Receptor: Structure–Activity Relationship Studies on 1-(4-Chlorophenyl)-3-{3-[6-(pyrrolidin-1-yl)pyridin-2-yl]phenyl}urea (PSNCBAM-1) JOURNAL ARTICLE published 25 September 2014 in Journal of Medicinal Chemistry Research funded by National Institute on Drug Abuse (DA003672,DA032837) |
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Synthesis, in Vitro Evaluation, and Radiolabeling of Fluorinated Puromycin Analogues: Potential Candidates for PET Imaging of Protein Synthesis JOURNAL ARTICLE published 27 October 2016 in Journal of Medicinal Chemistry Research funded by Medical Research Council (G9219778) |
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Discovery of Novel Tricyclic Full Agonists for the G-Protein-Coupled Niacin Receptor 109A with Minimized Flushing in Rats JOURNAL ARTICLE published 23 April 2009 in Journal of Medicinal Chemistry |
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Exploiting Protein Conformational Change to Optimize Adenosine-Derived Inhibitors of HSP70 JOURNAL ARTICLE published 26 May 2016 in Journal of Medicinal Chemistry Research funded by Cancer Research UK (C309/A11566,C309/A8274) |
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In VivoAnti-Chagas Vinylthio-, Vinylsulfinyl-, and Vinylsulfonylbenzofuroxan Derivatives JOURNAL ARTICLE published 1 November 2007 in Journal of Medicinal Chemistry |
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Synthesis and Structure−Activity Relationship Studies of 3,6-Diazabicyclo[3.2.0]heptanes as Novel α4β2 Nicotinic Acetylcholine Receptor Selective Agonists JOURNAL ARTICLE published 1 November 2007 in Journal of Medicinal Chemistry |
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Activity of Sulfonium Bisphosphonates on Tumor Cell Lines JOURNAL ARTICLE published 1 November 2007 in Journal of Medicinal Chemistry |
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Synthesis, Potency, and In Vivo Profiles of Quinoline Containing Histamine H3Receptor Inverse Agonists JOURNAL ARTICLE published 1 November 2007 in Journal of Medicinal Chemistry |
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Antiarrhythmic Hit to Lead Refinement in a Dish Using Patient-Derived iPSC Cardiomyocytes JOURNAL ARTICLE published 13 May 2021 in Journal of Medicinal Chemistry Research funded by California Institute for Regenerative Medicine (TR4-06857) |
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Design, Synthesis, and Multivariate Quantitative Structure−Activity Relationship of SalicylanilidesPotent Inhibitors of Type III Secretion inYersinia JOURNAL ARTICLE published 1 November 2007 in Journal of Medicinal Chemistry |
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Bifunctional and Unusual Amino Acid β- or γ-Ester Prodrugs of Nucleoside Analogues for Improved Affinity to ATB0,+ and Enhanced Metabolic Stability: An Application to Floxuridine JOURNAL ARTICLE published 8 October 2020 in Journal of Medicinal Chemistry Research funded by National Natural Science Foundation of China (81360485,81560577,81860630) | Natural Science Foundation of Jiangxi Province (20181BAB205087) | Key Project of Jiangxi (20192ACB70012) |
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Syntheses and Biological Activities (Topoisomerase Inhibition and Antitumor and Antimicrobial Properties) of Rebeccamycin Analogues Bearing Modified Sugar Moieties and Substituted on the Imide Nitrogen with a Methyl Group JOURNAL ARTICLE published 1 October 1997 in Journal of Medicinal Chemistry |