Metadata Search Funding Data Link References Status API Help
Facet browsing currently unavailable
Page 2 of 36494 results
Sort by: relevance publication year

Issue Publication Information

JOURNAL ARTICLE published 25 October 2018 in Journal of Medicinal Chemistry

Correction to A Novel Covalent mTOR Inhibitor, DHM25, Shows in Vivo Antitumor Activity against Triple-Negative Breast Cancer Cells

JOURNAL ARTICLE published 24 October 2019 in Journal of Medicinal Chemistry

Authors: Amélie Fouqué | Olivier Delalande | Mickael Jean | Rémy Castellano | Emmanuelle Josselin | Marine Malleter | Kenji F. Shoji | Mac Dinh Hung | Hariniaina Rampanarivo | Yves Collette | Pierre van de Weghe | Patrick Legembre

Issue Editorial Masthead

JOURNAL ARTICLE published 24 October 2019 in Journal of Medicinal Chemistry

Issue Publication Information

JOURNAL ARTICLE published 23 January 2020 in Journal of Medicinal Chemistry

Issue Publication Information

JOURNAL ARTICLE published 23 July 2020 in Journal of Medicinal Chemistry

Correction to “Discovery of the Bruton’s Tyrosine Kinase Inhibitor Clinical Candidate TAK-020 (S)-5-(1-((1-Acryloylpyrrolidin-3-yl)oxy)isoquinolin-3-yl)-2,4-dihydro-3H-1,2,4-triazol-3-one, by Fragment-Based Drug Design”

JOURNAL ARTICLE published 11 November 2021 in Journal of Medicinal Chemistry

Authors: Mark Sabat | Douglas R Dougan | Jacques Ermolieff | Petro Halkowycz | Beverly Knight | J. David Lawson | Nicholas Scorah | Christopher R Smith | Ewan R Taylor | Phong Vu | Corey Wyrick | Haixia Wang | Deepika Balakrishna | Mark Hixon | Loui Madakamutil | Donavon McConn

Issue Publication Information

JOURNAL ARTICLE published 10 January 2019 in Journal of Medicinal Chemistry

A Surprising Recipe for Designing Biased Ligands

JOURNAL ARTICLE published 10 January 2019 in Journal of Medicinal Chemistry

Authors: Sid Topiol

Issue Editorial Masthead

JOURNAL ARTICLE published 13 June 2019 in Journal of Medicinal Chemistry

Discovery of N-{4-[(3-Hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide Analogues as Selective Kappa Opioid Receptor Antagonists

JOURNAL ARTICLE published 13 June 2013 in Journal of Medicinal Chemistry

Authors: Chad M. Kormos | Chunyang Jin | Juan Pablo Cueva | Scott P. Runyon | James B. Thomas | Lawrence E. Brieaddy | S. Wayne Mascarella | Hernán A. Navarro | Brian P. Gilmour | F. Ivy Carroll

Issue Publication Information

JOURNAL ARTICLE published 14 July 2016 in Journal of Medicinal Chemistry

Antibody Recognition and Conformational Flexibility of a Plaque-Specific β-Amyloid Epitope Modulated by Non-native Peptide Flanking Regions

JOURNAL ARTICLE published 13 March 2008 in Journal of Medicinal Chemistry

Authors: Marilena Manea | Adrián Kalászi | Gábor Mező | Kata Horváti | Andrea Bodor | Anikó Horváth | Ödön Farkas | András Perczel | Michael Przybylski | Ferenc Hudecz

Antitumor Agents 260. New Desmosdumotin B Analogues with Improved In Vitro Anticancer Activity

JOURNAL ARTICLE published 1 June 2008 in Journal of Medicinal Chemistry

Authors: Kyoko Nakagawa-Goto | Kenneth F. Bastow | Tzu-Hsuan Chen | Susan L. Morris-Natschke | Kuo-Hsiung Lee

Design and Synthesis of a Series of l-trans-4-Substituted Prolines as Selective Antagonists for the Ionotropic Glutamate Receptors Including Functional and X-ray Crystallographic Studies of New Subtype Selective Kainic Acid Receptor Subtype 1 (GluK1) Antagonist (2S,4R)-4-(2-Carboxyphenoxy)pyrrolidine-2-carboxylic Acid

JOURNAL ARTICLE published 12 January 2017 in Journal of Medicinal Chemistry

Authors: Niels Krogsgaard-Larsen | Claudia G. Delgar | Karina Koch | Patricia M. G. E. Brown | Charlotte Møller | Liwei Han | Tri H. V. Huynh | Stinne W. Hansen | Birgitte Nielsen | Derek Bowie | Darryl S. Pickering | Jette Sandholm Kastrup | Karla Frydenvang | Lennart Bunch

blank page

JOURNAL ARTICLE published 1 December 1960 in Journal of Medicinal Chemistry

Benextramine-neuropeptide Y receptor interactions: contribution of the benzylic moieties to [3H]neuropeptide Y displacement activity

JOURNAL ARTICLE published January 1993 in Journal of Medicinal Chemistry

Authors: Michael B. Doughty | Chandra S. Chaurasia | Ke Li

Synthesis and 5-lipoxygenase inhibitory activities of eicosanoid compounds

JOURNAL ARTICLE published January 1983 in Journal of Medicinal Chemistry

Authors: Yoshinobu Arai | Katsuichi Shimoji | Mitoshi Konno | Yoshitaka Konishi | Shigehiro Okuyama | Sadahiko Iguchi | Masaki Hayashi | Tsumoru Miyamoto | Masaaki Toda

.pi.-Substituent constants for the 2H-1,2,4-benzothiadiazine 1,1-dioxide system

JOURNAL ARTICLE published April 1972 in Journal of Medicinal Chemistry

Authors: John G. Topliss | Milton D. Yudis

Folate analogs. 21. Synthesis and antifolate and antitumor activities of N10-(cyanomethyl)-5,8-dideazafolic acid

JOURNAL ARTICLE published April 1983 in Journal of Medicinal Chemistry

Authors: M. G. Nair | David C. Salter | R. L. Kisliuk | Y. Gaumont | G. North | F. M. Sirotnak

Antiviral compounds. 1. Structure-activity relationship of some antiviral enediones derived from aldehydo sugars

JOURNAL ARTICLE published January 1983 in Journal of Medicinal Chemistry

Authors: Eli Breuer | David Melumad | Shalom Sarel | Eva Margalith | Ehud Katz