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Showing results for ISSN matching 0022-2623

Preventive Oral Treatment with Resveratrol Pro-prodrugs Drastically Reduce Colon Inflammation in Rodents

JOURNAL ARTICLE published 28 October 2010 in Journal of Medicinal Chemistry

Authors: Mar Larrosa | Joao Tomé-Carneiro | María J. Yáñez-Gascón | David Alcántara | María V. Selma | David Beltrán | María T. García-Conesa | Cristina Urbán | Ricardo Lucas | Francisco Tomás-Barberán | Juan C. Morales | Juan Carlos Espín

https://doi.org/10.1021/jm1007006 Actions

Design, Synthesis, and Biological Evaluation of Monopyrrolinone-Based HIV-1 Protease Inhibitors

JOURNAL ARTICLE published 1 May 2003 in Journal of Medicinal Chemistry

Authors: Amos B. Smith | Louis-David Cantin | Alexander Pasternak | Lisa Guise-Zawacki | Wenquin Yao | Adam K. Charnley | Joseph Barbosa | Paul A. Sprengeler | Ralph Hirschmann | Sanjeev Munshi | David B. Olsen | William A. Schleif | Lawrence C. Kuo

https://doi.org/10.1021/jm0204587 Actions

Development of Novel Aminoglycoside (NB54) with Reduced Toxicity and Enhanced Suppression of Disease-Causing Premature Stop Mutations

JOURNAL ARTICLE published 14 May 2009 in Journal of Medicinal Chemistry

Authors: Igor Nudelman | Annie Rebibo-Sabbah | Marina Cherniavsky | Valery Belakhov | Mariana Hainrichson | Fuquan Chen | Jochen Schacht | Daniel S. Pilch | Tamar Ben-Yosef | Timor Baasov

https://doi.org/10.1021/jm801640k Actions

Design, Synthesis, and Antiviral Activity of Certain 2,5,6-Trihalo-1-(.beta.-D-ribofuranosyl)benzimidazoles

JOURNAL ARTICLE published September 1995 in Journal of Medicinal Chemistry

Authors: Leroy B. Townsend | Rodrigo V. Devivar | Steven R. Turk | M. Reza Nassiri | John C. Drach

https://doi.org/10.1021/jm00020a025 Actions

Synthesis and Anticancer Activity of Brefeldin A Ester Derivatives

JOURNAL ARTICLE published 1 June 2006 in Journal of Medicinal Chemistry

Authors: Nwanne O. Anadu | V. Jo Davisson | Mark Cushman

https://doi.org/10.1021/jm0602817 Actions

Structure−Activity Relationships of New 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as Allosteric Enhancers of the A3 Adenosine Receptor

JOURNAL ARTICLE published 1 June 2006 in Journal of Medicinal Chemistry

Authors: Anikó Göblyös | Zhan-Guo Gao | Johannes Brussee | Roberto Connestari | Sabrina Neves Santiago | Kai Ye | Adriaan P. IJzerman | Kenneth A. Jacobson

https://doi.org/10.1021/jm060086s Actions

Synthesis and Antiprotozoal Activity of N-Alkoxy Analogues of the Trypanocidal Lead Compound 4,4′-Bis(imidazolinylamino)diphenylamine with Improved Human Blood−Brain Barrier Permeability

JOURNAL ARTICLE published 27 January 2011 in Journal of Medicinal Chemistry

Authors: Lidia Nieto | Ainhoa Mascaraque | Florence Miller | Fabienne Glacial | Carlos Ríos Martínez | Marcel Kaiser | Reto Brun | Christophe Dardonville

https://doi.org/10.1021/jm101335q Actions

Enzyme-Activated Antagonists of the Strychnine-Insensitive Glycine/NMDA Receptor

JOURNAL ARTICLE published February 1994 in Journal of Medicinal Chemistry

Authors: Francesco G. Salituro | Ronald C. Tomlinson | Bruce M. Baron | Michael G. Palfreyman | Ian A. McDonald | Werner Schmidt | Hui Qiu Wu | Paolo Guidetti | Robert Schwarcz

https://doi.org/10.1021/jm00029a003 Actions

Synthesis and Characterization of an A6-A11 Methylene Thioacetal Human Insulin Analogue with Enhanced Stability

JOURNAL ARTICLE published 26 December 2019 in Journal of Medicinal Chemistry

Research funded by American Diabetes Association (#1-19-PDF110) | National Institute of Diabetes and Digestive and Kidney Diseases (R01DK120430)

Authors: Nan Zheng | Prasoona Karra | Michael A. VandenBerg | Jin Hwan Kim | Matthew J. Webber | William L. Holland | Danny Hung-Chieh Chou

https://doi.org/10.1021/acs.jmedchem.9b01589 Actions

Synthesis of (E)-5-(3,3,3-trifluoro-1-propenyl)-2'-deoxyuridine and related analogs: potent and unusually selective antiviral activity of (E)-5-(3,3,3-trifluoro-1-propenyl)-2'-deoxyridine against herpes simplex virus type 1

JOURNAL ARTICLE published March 1984 in Journal of Medicinal Chemistry

Authors: Donald E. Bergstrom | Jerry L. Ruth | P. Anantha Reddy | Erik De Clercq

https://doi.org/10.1021/jm00369a009 Actions

Novel Synthesis and Structural Characterization of a High-Affinity Paramagnetic Kinase Probe for the Identification of Non-ATP Site Binders by Nuclear Magnetic Resonance

JOURNAL ARTICLE published 11 February 2010 in Journal of Medicinal Chemistry

Authors: Franklin J. Moy | Arthur Lee | Lori Krim Gavrin | Zhang Bao Xu | Annette Sievers | Elizabeth Kieras | Wayne Stochaj | Lidia Mosyak | John McKew | Désirée H. H. Tsao

https://doi.org/10.1021/jm901525b Actions

Structure-Based Design, Synthesis, Evaluation, and Crystallographic Studies of Conformationally Constrained Smac Mimetics as Inhibitors of the X-linked Inhibitor of Apoptosis Protein (XIAP)

JOURNAL ARTICLE published 27 November 2008 in Journal of Medicinal Chemistry

Authors: Haiying Sun | Jeanne A. Stuckey | Zaneta Nikolovska-Coleska | Dongguang Qin | Jennifer L. Meagher | Su Qiu | Jianfeng Lu | Chao-Yie Yang | Naoyuki G. Saito | Shaomeng Wang

https://doi.org/10.1021/jm8006849 Actions

Effect of Chiral Purity on Adjuvanticity of Archaeol-Based Glycolipids

JOURNAL ARTICLE published 23 June 2022 in Journal of Medicinal Chemistry

Authors: Sophie Régnier | Edmond Lam | Vinicio Vasquez | Camilo F. Martinez-Farina | Felicity C. Stark | Gerard Agbayani | Lise Deschatelets | Renu Dudani | Blair A. Harrison | Bassel Akache | Michael J. McCluskie | Usha D. Hemraz

https://doi.org/10.1021/acs.jmedchem.2c00072 Actions

Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrimido[5,4-b]pyrrolizines as Novel Bruton’s Tyrosine Kinase Inhibitors

JOURNAL ARTICLE published 24 May 2018 in Journal of Medicinal Chemistry

Research funded by Government of Jiangsu Province (KYCX17_0684) | Science and Technology Commission of Shanghai Municipality (16XD1404600,14431900400) | National Natural Science Foundation of China (81703327,81773565,81430080) | Chinese Academy of Sciences (160621,GJHZ1622)

Authors: Yu Xue | Peiran Song | Zilan Song | Aoli Wang | Linjiang Tong | Meiyu Geng | Jian Ding | Qingsong Liu | Liping Sun | Hua Xie | Ao Zhang

https://doi.org/10.1021/acs.jmedchem.8b00441 Actions

Synthesis and Anticonvulsant Activity of Amino Acid-Derived Sulfamides

JOURNAL ARTICLE published 26 March 2009 in Journal of Medicinal Chemistry

Authors: Luciana Gavernet | Juan E. Elvira | Gisela A. Samaja | Valentina Pastore | Mariana Sella Cravero | Andrea Enrique | Guillermina Estiu | Luis E. Bruno-Blanch

https://doi.org/10.1021/jm800764p Actions

Subtype Selective Substrates for Histone Deacetylases

JOURNAL ARTICLE published 1 October 2004 in Journal of Medicinal Chemistry

Authors: Birgit Heltweg | Franck Dequiedt | Brett L. Marshall | Carsten Brauch | Minoru Yoshida | Norikazu Nishino | Eric Verdin | Manfred Jung

https://doi.org/10.1021/jm0497592 Actions

Synthesis, Structure−Activity Relationships, and Characterization of Novel Nonsteroidal and Selective Androgen Receptor Modulators

JOURNAL ARTICLE published 26 November 2009 in Journal of Medicinal Chemistry

Authors: Nathalie Schlienger | Birgitte W. Lund | Jan Pawlas | Fabrizio Badalassi | Fabio Bertozzi | Rasmus Lewinsky | Alma Fejzic | Mikkel B. Thygesen | Ali Tabatabaei | Stefania Risso Bradley | Luis R. Gardell | Fabrice Piu | Roger Olsson

https://doi.org/10.1021/jm901149c Actions

A Straightforward Approach for Engineering Efficacy and Selectivity at GPCRs

JOURNAL ARTICLE published 9 August 2012 in Journal of Medicinal Chemistry

Authors: Stefania Butini | Sandra Gemma | Giuseppe Campiani

https://doi.org/10.1021/jm301017v Actions

Issue Editorial Masthead

JOURNAL ARTICLE published 28 February 2019 in Journal of Medicinal Chemistry

https://doi.org/10.1021/jmv062i004_1261123 Actions

Corrections to Synthesis and Discovery of Water-Soluble Microtubule Targeting Agents that Bind to the Colchicine Site on Tubulin and Circumvent Pgp Mediated Resistance

JOURNAL ARTICLE published 10 February 2011 in Journal of Medicinal Chemistry

Authors: Aleem Gangjee | Ying Zhao | Lu Lin | Sudhir Raghavan | Elizabeth G. Roberts | April L. Risinger | Ernest Hamel | Susan L. Mooberry

https://doi.org/10.1021/jm101533s Actions
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